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Assay Detail

CHEMBL1007363

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Binding affinity to human SSTR2A
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Somatostatin receptor type 2 (CHEMBL1804)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

A synthetic method for peptide-PEG-lipid conjugates: application of octreotide-PEG-DSPE synthesis.
Su JC, Tseng CL, Chang TG, Yu WJ, Wu SK.
Bioorg Med Chem Lett (2008) 18 : 4593 -4596
PubMed 18656351 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 1 8.68 8.68

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL3350037 1 8.68

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL3350037 Ki = 2.1 nM 8.68