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Assay Detail

CHEMBL1007461

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Binding affinity to Escherichia coli 23S rRNA L11 binding domain
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Escherichia coli
Confidence 3 — Cell-line / Tissue
Curated By Autocuration

Target

Nucleic Acid (CHEMBL345)
Type NUCLEIC-ACID

Publication

Design and implementation of an ribonucleic acid (RNA) directed fragment library.
Bodoor K, Boyapati V, Gopu V, Boisdore M, Allam K, Miller J, Treleaven WD, Weldeghiorghis T, Aboul-ela F.
J Med Chem (2009) 52 : 3753 -3761
PubMed 19445516 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Kd 3 6.50 7.10

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL507798 MICROCOCCIN 1 7.10
CHEMBL1236460 THIOSTREPTON 1 5.89
CHEMBL2103750 NOSIHEPTIDE 2.0 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL507798 MICROCOCCIN Kd = 80.0 nM 7.10
CHEMBL1236460 THIOSTREPTON Kd = 1300.0 nM 5.89
CHEMBL2103750 NOSIHEPTIDE Kd < 3000.0 nM -