Assay Detail
ADMET
CHEMBL1007543
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Cytotoxicity against human NCI-H460 cells after 4 days by MTT assay
18
Total Activities
18
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | ADMET |
| Organism | Homo sapiens |
| Cell Type | NCI-H460 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Inhibition of staphyloxanthin virulence factor biosynthesis in Staphylococcus aureus: in vitro, in vivo, and crystallographic results.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 18 | 4.07 | 4.07 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL496803 | — | — | 1 | 4.07 |
| CHEMBL495623 | — | — | 1 | - |
| CHEMBL495624 | — | — | 1 | - |
| CHEMBL497634 | — | — | 1 | - |
| CHEMBL497635 | — | — | 1 | - |
| CHEMBL497616 | — | — | 1 | - |
| CHEMBL497617 | — | — | 1 | - |
| CHEMBL497815 | — | — | 1 | - |
| CHEMBL497410 | — | — | 1 | - |
| CHEMBL497618 | — | — | 1 | - |
| CHEMBL524084 | — | — | 1 | - |
| CHEMBL496801 | — | — | 1 | - |
| CHEMBL496802 | — | — | 1 | - |
| CHEMBL449115 | — | — | 1 | - |
| CHEMBL498628 | — | — | 1 | - |
| CHEMBL525377 | — | — | 1 | - |
| CHEMBL523897 | — | — | 1 | - |
| CHEMBL447414 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL496803 | — | IC50 | = | 86000.0 | nM | 4.07 |
| CHEMBL495623 | — | IC50 | > | 300000.0 | nM | - |
| CHEMBL495624 | — | IC50 | > | 300000.0 | nM | - |
| CHEMBL497634 | — | IC50 | > | 300000.0 | nM | - |
| CHEMBL497635 | — | IC50 | > | 300000.0 | nM | - |
| CHEMBL497616 | — | IC50 | > | 300000.0 | nM | - |
| CHEMBL497617 | — | IC50 | > | 300000.0 | nM | - |
| CHEMBL497815 | — | IC50 | > | 300000.0 | nM | - |
| CHEMBL497410 | — | IC50 | > | 300000.0 | nM | - |
| CHEMBL497618 | — | IC50 | > | 300000.0 | nM | - |
| CHEMBL524084 | — | IC50 | > | 300000.0 | nM | - |
| CHEMBL496801 | — | IC50 | > | 300000.0 | nM | - |
| CHEMBL496802 | — | IC50 | > | 300000.0 | nM | - |
| CHEMBL449115 | — | IC50 | = | 191000.0 | nM | - |
| CHEMBL498628 | — | IC50 | > | 300000.0 | nM | - |
| CHEMBL525377 | — | IC50 | = | 284000.0 | nM | - |
| CHEMBL523897 | — | IC50 | = | 306000.0 | nM | - |
| CHEMBL447414 | — | IC50 | > | 300000.0 | nM | - |