Assay Detail
Binding
CHEMBL1007903
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Binding affinity to OX2 receptor
18
Total Activities
18
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Intermediate |
Publication
Biomedical application of orexin/hypocretin receptor ligands in neuroscience.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 18 | 5.60 | 5.70 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL363743 | — | — | 1 | 5.70 |
| CHEMBL185136 | — | — | 1 | 5.60 |
| CHEMBL359632 | — | — | 1 | 5.50 |
| CHEMBL183786 | — | — | 1 | - |
| CHEMBL363951 | — | — | 1 | - |
| CHEMBL184384 | — | — | 1 | - |
| CHEMBL361748 | — | — | 1 | - |
| CHEMBL185435 | — | — | 1 | - |
| CHEMBL185382 | — | — | 1 | - |
| CHEMBL185219 | — | — | 1 | - |
| CHEMBL361716 | — | — | 1 | - |
| CHEMBL182473 | — | — | 1 | - |
| CHEMBL185093 | — | — | 1 | - |
| CHEMBL185088 | — | — | 1 | - |
| CHEMBL184936 | — | — | 1 | - |
| CHEMBL185080 | — | — | 1 | - |
| CHEMBL360377 | — | — | 1 | - |
| CHEMBL183576 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL363743 | — | Ki | = | 1995.26 | nM | 5.70 |
| CHEMBL185136 | — | Ki | = | 2511.89 | nM | 5.60 |
| CHEMBL359632 | — | Ki | = | 3162.28 | nM | 5.50 |
| CHEMBL183786 | — | Ki | > | 10000.0 | nM | - |
| CHEMBL363951 | — | Ki | > | 10000.0 | nM | - |
| CHEMBL184384 | — | Ki | > | 10000.0 | nM | - |
| CHEMBL361748 | — | Ki | > | 10000.0 | nM | - |
| CHEMBL185435 | — | Ki | > | 10000.0 | nM | - |
| CHEMBL185382 | — | Ki | > | 5011.87 | nM | - |
| CHEMBL185219 | — | Ki | > | 10000.0 | nM | - |
| CHEMBL361716 | — | Ki | > | 5011.87 | nM | - |
| CHEMBL182473 | — | Ki | > | 5011.87 | nM | - |
| CHEMBL185093 | — | Ki | > | 10000.0 | nM | - |
| CHEMBL185088 | — | Ki | > | 5011.87 | nM | - |
| CHEMBL184936 | — | Ki | > | 10000.0 | nM | - |
| CHEMBL185080 | — | Ki | > | 10000.0 | nM | - |
| CHEMBL360377 | — | Ki | > | 10000.0 | nM | - |
| CHEMBL183576 | — | Ki | > | 10000.0 | nM | - |