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Assay Detail

CHEMBL1008720

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Cytotoxicity against human HeLa cells by SRB assay
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type HeLa
Confidence 1 — Organism
Curated By Autocuration

Target

HeLa (CHEMBL399)
Type CELL-LINE
Organism Homo sapiens

Publication

Antitubercular sesterterpenes from the Thai sponge Brachiaster sp.
Wonganuchitmeta SN, Yuenyongsawad S, Keawpradub N, Plubrukarn A.
J Nat Prod (2004) 67 : 1767 -1770
PubMed 15497961 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 4 5.77 6.35

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL514498 HETERONEMIN 1 6.35
CHEMBL490765 1 5.78
CHEMBL250263 1 5.70
CHEMBL490567 1 5.26

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL514498 HETERONEMIN IC50 = 450.0 nM 6.35
CHEMBL490765 IC50 = 1680.0 nM 5.78
CHEMBL250263 IC50 = 1990.0 nM 5.70
CHEMBL490567 IC50 = 5490.0 nM 5.26