Assay Detail
Binding
CHEMBL1009869
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Binding affinity to CB1 receptor
5
Total Activities
5
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Intermediate |
Publication
Discovery of novel CB2 receptor ligands by a pharmacophore-based virtual screening workflow.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 5 | 5.72 | 6.42 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL498767 | — | — | 1 | 6.42 |
| CHEMBL371214 | — | — | 1 | 6.17 |
| CHEMBL73711 | — | — | 1 | 5.72 |
| CHEMBL408430 | — | — | 1 | 5.30 |
| CHEMBL497392 | — | — | 1 | 5.00 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL498767 | — | Ki | = | 381.0 | nM | 6.42 |
| CHEMBL371214 | — | Ki | = | 677.0 | nM | 6.17 |
| CHEMBL73711 | — | Ki | = | 1917.0 | nM | 5.72 |
| CHEMBL408430 | — | Ki | = | 5000.0 | nM | 5.30 |
| CHEMBL497392 | — | Ki | = | 10000.0 | nM | 5.00 |