Assay Detail
Binding
CHEMBL1010083
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Inhibition of Agrobacterium sp. beta galactosidase
7
Total Activities
7
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Agrobacterium sp. |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
1-Deoxygalactonojirimycin-lysine hybrids as potent D-galactosidase inhibitors.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 7 | 4.80 | 5.51 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL461161 | — | — | 1 | 5.51 |
| CHEMBL505422 | — | — | 1 | 5.00 |
| CHEMBL454920 | — | — | 1 | 4.68 |
| CHEMBL110458 | MIGALASTAT | 4.0 | 1 | 4.00 |
| CHEMBL459224 | — | — | 1 | - |
| CHEMBL508985 | — | — | 1 | - |
| CHEMBL446381 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL461161 | — | Ki | = | 3100.0 | nM | 5.51 |
| CHEMBL505422 | — | Ki | = | 10000.0 | nM | 5.00 |
| CHEMBL454920 | — | Ki | = | 21000.0 | nM | 4.68 |
| CHEMBL110458 | MIGALASTAT | Ki | = | 100000.0 | nM | 4.00 |
| CHEMBL459224 | — | Ki | = | 1900000.0 | nM | - |
| CHEMBL508985 | — | Ki | = | 170000.0 | nM | - |
| CHEMBL446381 | — | Ki | = | 140000.0 | nM | - |