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Assay Detail

CHEMBL1010560

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of HCV NS5B polymerase-mediated RNA synthesis
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Hepatitis C virus
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Target

Unchecked (CHEMBL612545)
Type UNCHECKED

Publication

The design, synthesis, and antiviral activity of monofluoro and difluoro analogues of 4'-azidocytidine against hepatitis C virus replication: the discovery of 4'-azido-2'-deoxy-2'-fluorocytidine and 4'-azido-2'-dideoxy-2',2'-difluorocytidine.
Smith DB, Kalayanov G, Sund C, Winqvist A, Maltseva T, Leveque VJ, Rajyaguru S, Le Pogam S, Najera I, Benkestock K, Zhou XX, Kaiser AC, Maag H, Cammack N, Martin JA, Swallow S, Johansson NG, Klumpp K, Smith M.
J Med Chem (2009) 52 : 2971 -2978
PubMed 19341305 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 1 5.89 5.89

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL393857 4'-AZIDOCYTIDINE -1.0 1 5.89

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL393857 4'-AZIDOCYTIDINE EC50 = 1280.0 nM 5.89