Assay Detail
Binding
CHEMBL1014326
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Binding affinity to mu opioid receptor in rhesus monkey brain membrane in absence of Na+ ions
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Macaca mulatta |
| Tissue | Brain |
| Subcellular | Membrane |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Ligand binding to nucleic acids and proteins: Does selectivity increase with strength?
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 1 | 10.70 | 10.70 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL312040 | ETONITAZENE | 2.0 | 1 | 10.70 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL312040 | ETONITAZENE | Ki | = | 0.02 | nM | 10.70 |