Assay Detail
Binding
CHEMBL1016980
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of EGF-stimulated RSK2 Ser386 autophosphorylation in serum starved african green monkey COS7 cells by immunoprecipitation and Western blot
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Chlorocebus aethiops |
| Cell Type | COS-7 |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Structural bioinformatics-based design of selective, irreversible kinase inhibitors.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 1 | 6.70 | 6.70 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL515414 | — | — | 1 | 6.70 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL515414 | — | EC50 | = | 200.0 | nM | 6.70 |