Assay Detail
Binding
CHEMBL1017392
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Binding affinity to vasopressin V1a receptor
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Intermediate |
Publication
Khusimol, a non-peptide ligand for vasopressin V1a receptors.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 7.58 | 8.70 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL419667 | RELCOVAPTAN | 2.0 | 1 | 8.70 |
| CHEMBL296908 | — | — | 1 | 6.46 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL419667 | RELCOVAPTAN | Ki | = | 2.0 | nM | 8.70 |
| CHEMBL296908 | — | Ki | = | 350.0 | nM | 6.46 |