Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL1034069

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Cytotoxicity against human SupT1 cells after 24 hrs by CellTiter-Blue assay
7
Total Activities
6
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type SUP-T1
Confidence 1 — Organism
Curated By Autocuration

Target

SUP-T1 (CHEMBL614940)
Type CELL-LINE
Organism Homo sapiens

Publication

Ceramides: branched alkyl chains in the sphingolipid siblings of diacylglycerol improve biological potency.
Kang JH, Garg H, Sigano DM, Francella N, Blumenthal R, Marquez VE.
Bioorg Med Chem (2009) 17 : 1498 -1505
PubMed 19171486 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 7 4.41 4.81

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL472237 1 4.81
CHEMBL471621 1 4.54
CHEMBL105867 2 4.38
CHEMBL224877 1 4.32
CHEMBL444967 1 4.28
CHEMBL471622 1 4.12

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL472237 IC50 = 15450.0 nM 4.81
CHEMBL471621 IC50 = 29080.0 nM 4.54
CHEMBL105867 IC50 = 41440.0 nM 4.38
CHEMBL224877 IC50 = 48010.0 nM 4.32
CHEMBL444967 IC50 = 52890.0 nM 4.28
CHEMBL471622 IC50 = 76300.0 nM 4.12
CHEMBL105867 IC50 > 200000.0 nM -