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Assay Detail

CHEMBL1034071

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Cytotoxicity against human MDA-MB-231 cells after 24 hrs by CellTiter-Blue assay
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type MDA-MB-231
Confidence 1 — Organism
Curated By Autocuration

Target

MDA-MB-231 (CHEMBL400)
Type CELL-LINE
Organism Homo sapiens

Publication

Ceramides: branched alkyl chains in the sphingolipid siblings of diacylglycerol improve biological potency.
Kang JH, Garg H, Sigano DM, Francella N, Blumenthal R, Marquez VE.
Bioorg Med Chem (2009) 17 : 1498 -1505
PubMed 19171486 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 2 4.55 4.65

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL472237 1 4.65
CHEMBL105867 1 4.45

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL472237 IC50 = 22360.0 nM 4.65
CHEMBL105867 IC50 = 35370.0 nM 4.45