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Assay Detail

CHEMBL1034188

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Functional
Antileishmanial activity against Leishmania donovani LV9 promastigotes after 96 hrs by MTT assay
7
Total Activities
7
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Leishmania donovani
Confidence 1 — Organism
Curated By Autocuration

Target

Leishmania donovani (CHEMBL367)
Type ORGANISM
Organism Leishmania donovani

Publication

Leishmanicidal and antiplasmodial activity of constituents of Smirnowia iranica.
Sairafianpour M, Kayser O, Christensen J, Asfa M, Witt M, Staerk D, Jaroszewski JW.
J Nat Prod (2002) 65 : 1754 -1758
PubMed 12502308 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 7 5.22 7.70

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL267345 AMPHOTERICIN B 4.0 1 7.70
CHEMBL501755 1 5.16
CHEMBL498724 SMIRANICIN 1 4.64
CHEMBL498725 GLYASPERIN H 1 4.60
CHEMBL454996 1 4.01
CHEMBL501754 1 -
CHEMBL489518 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL267345 AMPHOTERICIN B IC50 = 20.0 nM 7.70
CHEMBL501755 IC50 = 6900.0 nM 5.16
CHEMBL498724 SMIRANICIN IC50 = 22900.0 nM 4.64
CHEMBL498725 GLYASPERIN H IC50 = 25300.0 nM 4.60
CHEMBL454996 IC50 = 97000.0 nM 4.01
CHEMBL501754 IC50 = 232000.0 nM -
CHEMBL489518 IC50 = 395000.0 nM -