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Assay Detail

CHEMBL1039372

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of trypsin-activated human recombinant renin
30
Total Activities
30
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Renin (CHEMBL286)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Optimization of orally bioavailable alkyl amine renin inhibitors.
Xu Z, Cacatian S, Yuan J, Simpson RD, Jia L, Zhao W, Tice CM, Flaherty PT, Guo J, Ishchenko A, Singh SB, Wu Z, McKeever BM, Scott BB, Bukhtiyarov Y, Berbaum J, Mason J, Panemangalore R, Cappiello MG, Bentley R, Doe CP, Harrison RK, McGeehan GM, Dillard LW, Baldwin JJ, Claremon DA.
Bioorg Med Chem Lett (2010) 20 : 694 -699
PubMed 19959358 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 30 8.52 9.74

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL592763 1 9.74
CHEMBL589647 1 9.64
CHEMBL496430 1 9.33
CHEMBL591342 1 9.33
CHEMBL605408 1 9.32
CHEMBL591578 1 9.32
CHEMBL1639 ALISKIREN 4.0 1 9.28
CHEMBL592765 1 9.28
CHEMBL591340 1 9.24
CHEMBL592762 1 9.23
CHEMBL606238 1 9.21
CHEMBL590623 1 9.21
CHEMBL590388 1 9.21
CHEMBL591105 1 9.06
CHEMBL591341 1 8.93
CHEMBL589399 1 8.89
CHEMBL604248 1 8.82
CHEMBL590868 1 8.77
CHEMBL591104 1 8.68
CHEMBL590866 1 8.60
CHEMBL591579 1 7.85
CHEMBL608264 1 7.77
CHEMBL496416 1 7.68
CHEMBL592048 1 7.51
CHEMBL497821 1 7.40
CHEMBL591813 1 7.34
CHEMBL592047 1 7.34
CHEMBL606026 1 7.24
CHEMBL592284 1 6.75
CHEMBL591814 1 5.65

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL592763 IC50 = 0.18 nM 9.74
CHEMBL589647 IC50 = 0.23 nM 9.64
CHEMBL496430 IC50 = 0.47 nM 9.33
CHEMBL591342 IC50 = 0.47 nM 9.33
CHEMBL605408 IC50 = 0.48 nM 9.32
CHEMBL591578 IC50 = 0.48 nM 9.32
CHEMBL1639 ALISKIREN IC50 = 0.53 nM 9.28
CHEMBL592765 IC50 = 0.52 nM 9.28
CHEMBL591340 IC50 = 0.58 nM 9.24
CHEMBL592762 IC50 = 0.59 nM 9.23
CHEMBL606238 IC50 = 0.62 nM 9.21
CHEMBL590623 IC50 = 0.61 nM 9.21
CHEMBL590388 IC50 = 0.62 nM 9.21
CHEMBL591105 IC50 = 0.87 nM 9.06
CHEMBL591341 IC50 = 1.17 nM 8.93
CHEMBL589399 IC50 = 1.3 nM 8.89
CHEMBL604248 IC50 = 1.5 nM 8.82
CHEMBL590868 IC50 = 1.7 nM 8.77
CHEMBL591104 IC50 = 2.1 nM 8.68
CHEMBL590866 IC50 = 2.5 nM 8.60
CHEMBL591579 IC50 = 14.0 nM 7.85
CHEMBL608264 IC50 = 17.0 nM 7.77
CHEMBL496416 IC50 = 21.0 nM 7.68
CHEMBL592048 IC50 = 31.0 nM 7.51
CHEMBL497821 IC50 = 40.0 nM 7.40
CHEMBL591813 IC50 = 46.0 nM 7.34
CHEMBL592047 IC50 = 46.0 nM 7.34
CHEMBL606026 IC50 = 57.0 nM 7.24
CHEMBL592284 IC50 = 177.0 nM 6.75
CHEMBL591814 IC50 = 2260.0 nM 5.65