Assay Detail
Binding
CHEMBL1041297
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Inhibition of VIM2 using nitrocefin as substrate by rapid dilution method
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Inhibitors of VIM-2 by screening pharmacologically active and click-chemistry compound libraries.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 3 | 6.02 | 6.39 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL578035 | — | — | 1 | 6.39 |
| CHEMBL584206 | — | — | 1 | 5.85 |
| CHEMBL58 | MITOXANTRONE | 4.0 | 1 | 5.82 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL578035 | — | Ki | = | 410.0 | nM | 6.39 |
| CHEMBL584206 | — | Ki | = | 1410.0 | nM | 5.85 |
| CHEMBL58 | MITOXANTRONE | Ki | = | 1500.0 | nM | 5.82 |