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Assay Detail

CHEMBL1045653

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Functional
Antiproliferative activity against mouse L1210 cells
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Mus musculus
Cell Type L1210
Confidence 1 — Organism
Curated By Autocuration

Target

L1210 (CHEMBL386)
Type CELL-LINE
Organism Mus musculus

Publication

Thiosemicarbazones from the old to new: iron chelators that are more than just ribonucleotide reductase inhibitors.
Yu Y, Kalinowski DS, Kovacevic Z, Siafakas AR, Jansson PJ, Stefani C, Lovejoy DB, Sharpe PC, Bernhardt PV, Richardson DR, Richardson DR.
J Med Chem (2009) 52 : 5271 -5294
PubMed 19601577 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 2 5.48 6.70

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL70927 DEFERIPRONE 4.0 1 6.70
CHEMBL150911 1 4.26

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL70927 DEFERIPRONE IC50 = 200.0 nM 6.70
CHEMBL150911 IC50 = 55000.0 nM 4.26