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Assay Detail

CHEMBL1050384

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Binding affinity to ghrelin receptor
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Confidence 8 — Homologous single protein target
Curated By Autocuration

Target

Growth hormone secretagogue receptor type 1 (CHEMBL4616)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Triazole oxytocin antagonists: Identification of an aryloxyazetidine replacement for a biaryl substituent.
Brown A, Brown TB, Calabrese A, Ellis D, Puhalo N, Ralph M, Watson L.
Bioorg Med Chem Lett (2010) 20 : 516 -520
PubMed 19963374 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 1 5.36 5.36

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL594828 1 5.36

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL594828 Ki = 4400.0 nM 5.36