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Assay Detail

CHEMBL1052303

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiviral activity against HCV1b BK infected in human H2B2 cells expressing HEPREP 2b replicon by cell-ELISA assay
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Hepacivirus hominis
Cell Type H2B2
Confidence 1 — Organism
Curated By Autocuration

Target

Hepatitis C virus (CHEMBL379)
Type ORGANISM
Organism Hepacivirus hominis

Publication

Identification and biological evaluation of a series of 1H-benzo[de]isoquinoline-1,3(2H)-diones as hepatitis C virus NS5B polymerase inhibitors.
Ontoria JM, Rydberg EH, Di Marco S, Tomei L, Attenni B, Malancona S, Martin Hernando JI, Gennari N, Koch U, Narjes F, Rowley M, Summa V, Carroll SS, Olsen DB, De Francesco R, Altamura S, Migliaccio G, Carfì A.
J Med Chem (2009) 52 : 5217 -5227
PubMed 19877603 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 1 4.96 4.96

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL559638 1 4.96

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL559638 EC50 = 11000.0 nM 4.96