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Assay Detail

CHEMBL1060746

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of dog EP3 receptor
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Canis lupus familiaris
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Target

Unchecked (CHEMBL612545)
Type UNCHECKED

Publication

Discovery of novel aminothiadiazole amides as selective EP(3) receptor antagonists.
Hilfiker MA, Wang N, Hou X, Du Z, Pullen MA, Nord M, Nagilla R, Fries HE, Wu CW, Sulpizio AC, Jaworski JP, Morrow D, Edwards RM, Jin J.
Bioorg Med Chem Lett (2009) 19 : 4292 -4295
PubMed 19487124 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 1 7.90 7.90

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL563480 1 7.90

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL563480 EC50 = 12.59 nM 7.90