Assay Detail
Binding
CHEMBL1061191
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of AMPK in the presence of 50uM ATP
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Rattus norvegicus |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
The selectivity of protein kinase inhibitors: a further update.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 6.88 | 6.96 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL605003 | — | — | 1 | 6.96 |
| CHEMBL265470 | — | — | 1 | 6.80 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL605003 | — | IC50 | = | 110.0 | nM | 6.96 |
| CHEMBL265470 | — | IC50 | = | 160.0 | nM | 6.80 |