Assay Detail
Binding
CHEMBL1061990
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Inhibition of BRSK2 in the presence of 50uM ATP
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Expert |
Target
Serine/threonine-protein kinase BRSK2 (CHEMBL4574) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
The selectivity of protein kinase inhibitors: a further update.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 6.48 | 7.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL605003 | — | — | 1 | 7.00 |
| CHEMBL1240885 | — | — | 1 | 5.96 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL605003 | — | IC50 | = | 100.0 | nM | 7.00 |
| CHEMBL1240885 | — | IC50 | = | 1100.0 | nM | 5.96 |