Assay Detail
Binding
CHEMBL1065678
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of rat NTPdase3 by capillary electrophoresis method
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Rattus norvegicus |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Nucleoside triphosphate diphosphohydrolase 3 (CHEMBL1075237) ↗| Type | SINGLE PROTEIN |
| Organism | Rattus norvegicus |
Publication
Development of potent and selective inhibitors of ecto-5'-nucleotidase based on an anthraquinone scaffold.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 4 | 5.54 | 5.96 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL223344 | RB 2 | — | 1 | 5.96 |
| CHEMBL498423 | — | — | 1 | 5.82 |
| CHEMBL256057 | ACID BLUE 25 | — | 1 | 4.84 |
| CHEMBL496030 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL223344 | RB 2 | Ki | = | 1100.0 | nM | 5.96 |
| CHEMBL498423 | — | Ki | = | 1500.0 | nM | 5.82 |
| CHEMBL256057 | ACID BLUE 25 | Ki | = | 14300.0 | nM | 4.84 |
| CHEMBL496030 | — | Ki | - | — | - |