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Assay Detail

CHEMBL1067221

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of Dengue virus type 2 NS5 RNA methyltransferase at 80 nM enzyme concentration
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism dengue virus type 2
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Genome polyprotein (CHEMBL3308998)
Type SINGLE PROTEIN
Organism dengue virus type 2

Publication

Novel inhibitors of dengue virus methyltransferase: discovery by in vitro-driven virtual screening on a desktop computer grid.
Podvinec M, Lim SP, Schmidt T, Scarsi M, Wen D, Sonntag LS, Sanschagrin P, Shenkin PS, Schwede T.
J Med Chem (2010) 53 : 1483 -1495
PubMed 20108931 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 2 5.07 5.15

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL115145 1 5.15
CHEMBL597979 1 4.99

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL115145 IC50 = 7140.0 nM 5.15
CHEMBL597979 IC50 = 10240.0 nM 4.99