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Assay Detail

CHEMBL1067226

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Binding
Inhibition of recombinant wild type HIV1 protease assessed as hydrolysis of fluorogenic substrate
12
Total Activities
12
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Human immunodeficiency virus 1
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Protease (CHEMBL2366517)
Type SINGLE PROTEIN
Organism Human immunodeficiency virus 1

Publication

Synthesis of new thienyl ring containing HIV-1 protease inhibitors: promising preliminary pharmacological evaluation against recombinant HIV-1 proteases.
Bonini C, Chiummiento L, De Bonis M, Di Blasio N, Funicello M, Lupattelli P, Pandolfo R, Tramutola F, Berti F.
J Med Chem (2010) 53 : 1451 -1457
PubMed 20108932 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 12 7.46 9.40

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL114 SAQUINAVIR 4.0 1 9.40
CHEMBL591934 1 9.22
CHEMBL577443 1 8.92
CHEMBL584 NELFINAVIR 4.0 1 8.72
CHEMBL606392 1 8.54
CHEMBL577638 1 8.22
CHEMBL591933 1 7.82
CHEMBL578278 1 7.68
CHEMBL578874 1 5.82
CHEMBL578053 1 5.40
CHEMBL577017 1 5.30
CHEMBL597982 1 4.52

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL114 SAQUINAVIR IC50 = 0.4 nM 9.40
CHEMBL591934 IC50 = 0.6 nM 9.22
CHEMBL577443 IC50 = 1.2 nM 8.92
CHEMBL584 NELFINAVIR IC50 = 1.9 nM 8.72
CHEMBL606392 IC50 = 2.9 nM 8.54
CHEMBL577638 IC50 = 6.0 nM 8.22
CHEMBL591933 IC50 = 15.0 nM 7.82
CHEMBL578278 IC50 = 21.0 nM 7.68
CHEMBL578874 IC50 = 1500.0 nM 5.82
CHEMBL578053 IC50 = 4000.0 nM 5.40
CHEMBL577017 IC50 = 5000.0 nM 5.30
CHEMBL597982 IC50 = 30000.0 nM 4.52