Assay Detail
Functional
CHEMBL1067693
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Agonist activity at P2Y1 receptor expressed in human HEK293 cells
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Cell Type | HEK293 |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
A novel insulin secretagogue based on a dinucleoside polyphosphate scaffold.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 2 | 7.65 | 8.59 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2309024 | — | — | 1 | 8.59 |
| CHEMBL14249 | ADENOSINE TRIPHOSPHATE | 2.0 | 1 | 6.70 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2309024 | — | EC50 | = | 2.6 | nM | 8.59 |
| CHEMBL14249 | ADENOSINE TRIPHOSPHATE | EC50 | = | 200.0 | nM | 6.70 |