Assay Detail
Binding
CHEMBL1072176
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Displacement of [3H]5CT from 5HT7B receptor
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
SAR studies on new bis-aryls 5-HT7 ligands: Synthesis and molecular modeling.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 8.81 | 9.22 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL161765 | — | — | 1 | 9.22 |
| CHEMBL158285 | — | — | 1 | 8.39 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL161765 | — | Ki | = | 0.6 | nM | 9.22 |
| CHEMBL158285 | — | Ki | = | 4.1 | nM | 8.39 |