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Assay Detail

CHEMBL1101679

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiviral activity against Vesicular stomatitis virus infected in EPT cells assessed as inhibition of virus-induced cytopathic effect treated immediately after viral infection measured after 24 hrs
12
Total Activities
12
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Vesicular stomatitis virus
Cell Type EPT
Confidence 1 — Organism
Curated By Autocuration

Target

Vesicular stomatitis virus (CHEMBL613739)
Type ORGANISM
Organism Vesicular stomatitis virus

Publication

Synthesis, cytotoxicity, antiviral activity and interferon inducing ability of 6-(2-aminoethyl)-6H-indolo[2,3-b]quinoxalines.
Shibinskaya MO, Lyakhov SA, Mazepa AV, Andronati SA, Turov AV, Zholobak NM, Spivak NY.
Eur J Med Chem (2010) 45 : 1237 -1243
PubMed 20056519 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 12 5.14 5.39

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1088346 1 5.39
CHEMBL1098690 1 5.39
CHEMBL1084906 1 5.33
CHEMBL1098374 1 5.32
CHEMBL1098691 1 5.25
CHEMBL1092508 1 5.21
CHEMBL1077006 1 5.18
CHEMBL1084905 1 5.10
CHEMBL1092507 1 5.02
CHEMBL1098689 1 4.88
CHEMBL539581 TILORONE HYDROCHLORIDE -1.0 1 4.87
CHEMBL1088347 1 4.70

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1088346 IC50 = 4073.8 nM 5.39
CHEMBL1098690 IC50 = 4073.8 nM 5.39
CHEMBL1084906 IC50 = 4677.35 nM 5.33
CHEMBL1098374 IC50 = 4786.3 nM 5.32
CHEMBL1098691 IC50 = 5623.41 nM 5.25
CHEMBL1092508 IC50 = 6165.95 nM 5.21
CHEMBL1077006 IC50 = 6606.93 nM 5.18
CHEMBL1084905 IC50 = 7943.28 nM 5.10
CHEMBL1092507 IC50 = 9549.93 nM 5.02
CHEMBL1098689 IC50 = 13182.57 nM 4.88
CHEMBL539581 TILORONE HYDROCHLORIDE IC50 = 13489.63 nM 4.87
CHEMBL1088347 IC50 = 19952.62 nM 4.70