Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL1102995

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of CDK3
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Confidence 8 — Homologous single protein target
Curated By Autocuration

Target

Cyclin-dependent kinase 3 (CHEMBL4442)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Discovery of potent and bioavailable GSK-3beta inhibitors.
Gong L, Hirschfeld D, Tan YC, Heather Hogg J, Peltz G, Avnur Z, Dunten P.
Bioorg Med Chem Lett (2010) 20 : 1693 -1696
PubMed 20138512 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Kd 1 7.10 7.10

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1082152 1 7.10

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1082152 Kd = 80.0 nM 7.10