Assay Detail
Functional
CHEMBL1107394
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Antagonist activity at P2Y12 receptor by [35S]GTPgammaS binding assay
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Frontal affinity chromatography-mass spectrometry useful for characterization of new ligands for GPR17 receptor.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 9.15 | 9.15 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1097279 | CANGRELOR TETRASODIUM | 4.0 | 1 | 9.15 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1097279 | CANGRELOR TETRASODIUM | IC50 | = | 0.7 | nM | 9.15 |