Assay Detail
Binding
CHEMBL1107839
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of human Integrin alpha5beta3 receptors expressed in HOP cells assessed as cell attachment after 30 mins by colorimetric assay
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Cell Type | HOP |
| Confidence | 7 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Ultrasmall particle of iron oxide--RGD peptidomimetic conjugate: synthesis and characterisation.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 3 | 9.56 | 10.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL565693 | — | — | 1 | 10.00 |
| CHEMBL1077192 | — | — | 1 | 9.52 |
| CHEMBL1077191 | — | — | 1 | 9.15 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL565693 | — | IC50 | = | 0.1 | nM | 10.00 |
| CHEMBL1077192 | — | IC50 | = | 0.3 | nM | 9.52 |
| CHEMBL1077191 | — | IC50 | = | 0.7 | nM | 9.15 |