Assay Detail
Binding
CHEMBL1108470
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Inhibition of JNK1 by high throughput screening
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
1-Aryl-3,4-dihydroisoquinoline inhibitors of JNK3.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 6.75 | 7.10 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL194806 | — | — | 1 | 7.10 |
| CHEMBL203535 | — | — | 1 | 6.40 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL194806 | — | IC50 | = | 79.43 | nM | 7.10 |
| CHEMBL203535 | — | IC50 | = | 398.11 | nM | 6.40 |