Assay Detail
Binding
CHEMBL1110133
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of recombinant DPP4
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Inhibitors of prolyl oligopeptidases for the therapy of human diseases: defining diseases and inhibitors.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 5.72 | 6.42 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL217561 | — | — | 1 | 6.42 |
| CHEMBL386890 | — | — | 1 | 5.02 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL217561 | — | Ki | = | 377.0 | nM | 6.42 |
| CHEMBL386890 | — | Ki | = | 9500.0 | nM | 5.02 |