Assay Detail
Binding
CHEMBL1114459
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Inhibition of IgG binding to soluble human FcRn after 5 hrs by competition ELISA
30
Total Activities
30
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Synthesis and structure-activity relationships of dimeric peptide antagonists of the human immunoglobulin G-human neonatal Fc receptor (IgG-FcRn) interaction.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 30 | 7.06 | 8.80 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1090633 | — | — | 1 | 8.80 |
| CHEMBL1090970 | — | — | 1 | 8.62 |
| CHEMBL1090632 | — | — | 1 | 8.62 |
| CHEMBL2304309 | — | — | 1 | 8.59 |
| CHEMBL1090640 | — | — | 1 | 8.41 |
| CHEMBL1090278 | — | — | 1 | 8.41 |
| CHEMBL1090968 | — | — | 1 | 8.38 |
| CHEMBL1090638 | — | — | 1 | 8.34 |
| CHEMBL1090636 | — | — | 1 | 8.33 |
| CHEMBL2304310 | — | — | 1 | 8.32 |
| CHEMBL1090637 | — | — | 1 | 8.30 |
| CHEMBL1090635 | — | — | 1 | 8.28 |
| CHEMBL1090639 | — | — | 1 | 8.25 |
| CHEMBL1090279 | — | — | 1 | 7.75 |
| CHEMBL1090969 | — | — | 1 | 7.70 |
| CHEMBL1090280 | — | — | 1 | 7.30 |
| CHEMBL1089946 | — | — | 1 | 6.37 |
| CHEMBL1089948 | — | — | 1 | 6.28 |
| CHEMBL1090276 | — | — | 1 | 6.24 |
| CHEMBL1089952 | — | — | 1 | 6.22 |
| CHEMBL1090275 | — | — | 1 | 6.15 |
| CHEMBL1089949 | — | — | 1 | 6.00 |
| CHEMBL1090274 | — | — | 1 | 5.96 |
| CHEMBL1089947 | — | — | 1 | 5.96 |
| CHEMBL2304308 | — | — | 1 | 5.72 |
| CHEMBL1090273 | — | — | 1 | 5.62 |
| CHEMBL1090277 | — | — | 1 | 5.52 |
| CHEMBL1089950 | — | — | 1 | 4.66 |
| CHEMBL1089945 | — | — | 1 | 4.43 |
| CHEMBL1089944 | — | — | 1 | 4.40 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1090633 | — | IC50 | = | 1.6 | nM | 8.80 |
| CHEMBL1090970 | — | IC50 | = | 2.4 | nM | 8.62 |
| CHEMBL1090632 | — | IC50 | = | 2.4 | nM | 8.62 |
| CHEMBL2304309 | — | IC50 | = | 2.6 | nM | 8.59 |
| CHEMBL1090640 | — | IC50 | = | 3.9 | nM | 8.41 |
| CHEMBL1090278 | — | IC50 | = | 3.9 | nM | 8.41 |
| CHEMBL1090968 | — | IC50 | = | 4.2 | nM | 8.38 |
| CHEMBL1090638 | — | IC50 | = | 4.6 | nM | 8.34 |
| CHEMBL1090636 | — | IC50 | = | 4.7 | nM | 8.33 |
| CHEMBL2304310 | — | IC50 | = | 4.8 | nM | 8.32 |
| CHEMBL1090637 | — | IC50 | = | 5.0 | nM | 8.30 |
| CHEMBL1090635 | — | IC50 | = | 5.2 | nM | 8.28 |
| CHEMBL1090639 | — | IC50 | = | 5.6 | nM | 8.25 |
| CHEMBL1090279 | — | IC50 | = | 18.0 | nM | 7.75 |
| CHEMBL1090969 | — | IC50 | = | 20.0 | nM | 7.70 |
| CHEMBL1090280 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL1089946 | — | IC50 | = | 430.0 | nM | 6.37 |
| CHEMBL1089948 | — | IC50 | = | 520.0 | nM | 6.28 |
| CHEMBL1090276 | — | IC50 | = | 580.0 | nM | 6.24 |
| CHEMBL1089952 | — | IC50 | = | 600.0 | nM | 6.22 |
| CHEMBL1090275 | — | IC50 | = | 710.0 | nM | 6.15 |
| CHEMBL1089949 | — | IC50 | = | 1000.0 | nM | 6.00 |
| CHEMBL1090274 | — | IC50 | = | 1100.0 | nM | 5.96 |
| CHEMBL1089947 | — | IC50 | = | 1100.0 | nM | 5.96 |
| CHEMBL2304308 | — | IC50 | = | 1900.0 | nM | 5.72 |
| CHEMBL1090273 | — | IC50 | = | 2400.0 | nM | 5.62 |
| CHEMBL1090277 | — | IC50 | = | 3000.0 | nM | 5.52 |
| CHEMBL1089950 | — | IC50 | = | 22000.0 | nM | 4.66 |
| CHEMBL1089945 | — | IC50 | = | 37000.0 | nM | 4.43 |
| CHEMBL1089944 | — | IC50 | = | 40000.0 | nM | 4.40 |