Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL1115069

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Inhibition of HCV 1b NS5B Cdelta21 RNA dependent RNA polymerase expressed in Escherichia coli after 30 mins by fluorescence assay
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Hepatitis C virus subtype 1b
Confidence 1 — Organism
Curated By Autocuration

Target

Hepatitis C virus (CHEMBL379)
Type ORGANISM
Organism Hepacivirus hominis

Publication

Antiviral activity of benzimidazole derivatives. II. Antiviral activity of 2-phenylbenzimidazole derivatives.
Tonelli M, Simone M, Tasso B, Novelli F, Boido V, Sparatore F, Paglietti G, Pricl S, Giliberti G, Blois S, Ibba C, Sanna G, Loddo R, La Colla P.
Bioorg Med Chem (2010) 18 : 2937 -2953
PubMed 20359898 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 3 4.77 5.30

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1093511 1 5.30
CHEMBL1088991 1 4.52
CHEMBL159895 1 4.48

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1093511 IC50 = 5000.0 nM 5.30
CHEMBL1088991 IC50 = 30000.0 nM 4.52
CHEMBL159895 IC50 = 33000.0 nM 4.48