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Assay Detail

CHEMBL1118889

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Binding
Inhibition of MMP2
30
Total Activities
30
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Confidence 8 — Homologous single protein target
Curated By Autocuration

Target

72 kDa type IV collagenase (CHEMBL333)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Orally bioavailable dual MMP-1/MMP-14 sparing, MMP-13 selective alpha-sulfone hydroxamates.
Kolodziej SA, Hockerman SL, Boehm TL, Carroll JN, DeCrescenzo GA, McDonald JJ, Mischke DA, Munie GE, Fletcher TR, Rico JG, Stehle NW, Swearingen C, Becker DP.
Bioorg Med Chem Lett (2010) 20 : 3557 -3560
PubMed 20529684 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 30 7.07 9.48

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1082381 1 9.48
CHEMBL1084221 1 8.70
CHEMBL1084509 1 8.43
CHEMBL1083932 1 8.36
CHEMBL1084510 1 8.28
CHEMBL1084218 1 8.27
CHEMBL1084238 1 7.92
CHEMBL1084208 1 7.74
CHEMBL1082966 1 7.68
CHEMBL1085602 1 7.63
CHEMBL1083931 1 7.49
CHEMBL1084209 1 7.46
CHEMBL1083907 1 7.40
CHEMBL1084206 1 7.31
CHEMBL1083322 1 7.16
CHEMBL1083625 1 7.09
CHEMBL1083906 1 7.06
CHEMBL1084207 1 6.48
CHEMBL1083908 1 6.43
CHEMBL1082370 1 6.30
CHEMBL1082371 1 6.30
CHEMBL1083626 1 6.16
CHEMBL1085264 1 6.10
CHEMBL1083007 1 6.05
CHEMBL1084217 1 5.85
CHEMBL1085263 1 5.76
CHEMBL1083321 1 5.51
CHEMBL1084220 1 5.43
CHEMBL1085988 1 5.27
CHEMBL1085748 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1082381 IC50 = 0.33 nM 9.48
CHEMBL1084221 IC50 = 2.0 nM 8.70
CHEMBL1084509 IC50 = 3.7 nM 8.43
CHEMBL1083932 IC50 = 4.4 nM 8.36
CHEMBL1084510 IC50 = 5.3 nM 8.28
CHEMBL1084218 IC50 = 5.4 nM 8.27
CHEMBL1084238 IC50 = 12.1 nM 7.92
CHEMBL1084208 IC50 = 18.4 nM 7.74
CHEMBL1082966 IC50 = 21.1 nM 7.68
CHEMBL1085602 IC50 = 23.5 nM 7.63
CHEMBL1083931 IC50 = 32.6 nM 7.49
CHEMBL1084209 IC50 = 35.0 nM 7.46
CHEMBL1083907 IC50 = 40.0 nM 7.40
CHEMBL1084206 IC50 = 48.5 nM 7.31
CHEMBL1083322 IC50 = 70.0 nM 7.16
CHEMBL1083625 IC50 = 82.0 nM 7.09
CHEMBL1083906 IC50 = 88.0 nM 7.06
CHEMBL1084207 IC50 = 330.0 nM 6.48
CHEMBL1083908 IC50 = 370.0 nM 6.43
CHEMBL1082370 IC50 = 500.0 nM 6.30
CHEMBL1082371 IC50 = 505.0 nM 6.30
CHEMBL1083626 IC50 = 700.0 nM 6.16
CHEMBL1085264 IC50 = 800.0 nM 6.10
CHEMBL1083007 IC50 = 900.0 nM 6.05
CHEMBL1084217 IC50 = 1400.0 nM 5.85
CHEMBL1085263 IC50 = 1750.0 nM 5.76
CHEMBL1083321 IC50 = 3100.0 nM 5.51
CHEMBL1084220 IC50 = 3700.0 nM 5.43
CHEMBL1085988 IC50 = 5400.0 nM 5.27
CHEMBL1085748 IC50 > 10000.0 nM -