Assay Detail
Binding
CHEMBL1120076
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Displacement of 8-anilino-1-naphthalene-sulfonic acid from human FABP4 F16A mutant expressed in Escherichia coli BL21 (DE3) cells after 3 mins
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Cell Type | BL21-DE3 |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Discovery of highly selective inhibitors of human fatty acid binding protein 4 (FABP4) by virtual screening.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 3 | 4.12 | 4.12 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1085571 | — | — | 1 | 4.12 |
| CHEMBL1085570 | — | — | 1 | - |
| CHEMBL267476 | LINOLEIC ACID | 2.0 | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1085571 | — | IC50 | = | 76500.0 | nM | 4.12 |
| CHEMBL1085570 | — | IC50 | - | — | - | |
| CHEMBL267476 | LINOLEIC ACID | IC50 | - | — | - |