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Assay Detail

CHEMBL1120702

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Binding affinity to EP3 receptor
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Confidence 8 — Homologous single protein target
Curated By Autocuration

Target

Prostaglandin E2 receptor EP3 subtype (CHEMBL3710)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Emerging targets in osteoporosis disease modification.
Allen JG, Fotsch C, Babij P.
J Med Chem (2010) 53 : 4332 -4353
PubMed 20218623 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 9.03 9.03

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL548 DINOPROSTONE 4.0 1 9.03

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL548 DINOPROSTONE IC50 = 0.94 nM 9.03