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Assay Detail

CHEMBL1166153

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Binding
Inhibition of Saccharomyces cerevisiae uridine 5'-monophosphate synthase after overnight incubation at room temperature by VP-ITC microcalorimetry
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Saccharomyces cerevisiae
Confidence 8 — Homologous single protein target
Curated By Autocuration

Target

Orotidine 5'-phosphate decarboxylase (CHEMBL4858)
Type SINGLE PROTEIN
Organism Saccharomyces cerevisiae S288c

Publication

Structural determinants for the inhibitory ligands of orotidine-5'-monophosphate decarboxylase.
Meza-Avina ME, Wei L, Liu Y, Poduch E, Bello AM, Mishra RK, Pai EF, Kotra LP.
Bioorg Med Chem (2010) 18 : 4032 -4041
PubMed 20452222 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 2 8.30 8.30

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1164953 1 8.30
CHEMBL383923 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1164953 Ki = 5.0 nM 8.30
CHEMBL383923 Ki = 0.009 nM -