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Assay Detail

CHEMBL1168035

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of rice alpha-glucosidase assessed as D-glucose release at pH 5 after 10 to 30 mins
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Oryza sativa
Confidence 8 — Homologous single protein target
Curated By Autocuration

Target

Probable alpha-glucosidase Os06g0675700 (CHEMBL1163102)
Type SINGLE PROTEIN
Organism Oryza sativa Japonica Group

Publication

2,5-Dideoxy-2,5-imino-d-altritol as a new class of pharmacological chaperone for Fabry disease.
Kato A, Yamashita Y, Nakagawa S, Koike Y, Adachi I, Hollinshead J, Nash RJ, Ikeda K, Asano N.
Bioorg Med Chem (2010) 18 : 3790 -3794
PubMed 20457528 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 4 4.68 5.00

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1163255 1 5.00
CHEMBL1163562 1 4.35
CHEMBL469844 1 -
CHEMBL1163254 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1163255 IC50 = 10000.0 nM 5.00
CHEMBL1163562 IC50 = 45000.0 nM 4.35
CHEMBL469844 IC50 = 171000.0 nM -
CHEMBL1163254 IC50 = 670000.0 nM -