Assay Detail

CHEMBL1217090

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding

Inhibition of Plasmodium falciparum protein farnesyltransferase

ChEMBL ↗

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Target

Unchecked (CHEMBL612545) ↗

Open DB target context

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Primary target Unchecked

CHEMBL612545

Anchored from Assay target.

Protein identity Unchecked

Disease frame Disease evidence pending

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Review focus Open DB context pending

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Total Activities

Compounds Tested

Activity Types

Assay Parameters

Assay Information

Assay Type	Binding
Organism	Plasmodium falciparum
Confidence	0 — Uncurated / Unknown
Curated By	Autocuration

Target

Unchecked (CHEMBL612545) ↗

Type

UNCHECKED

Publication

Quinolines and structurally related heterocycles as antimalarials.

Kaur K, Jain M, Reddy RP, Jain R.
Eur J Med Chem (2010) 45 : 3245 -3264
PubMed 20466465 · DOI

Activity Statistics

Type	Count	Avg pChEMBL	Best pChEMBL
IC50	1	9.22	9.22

Compounds Tested

Compound	Name	Phase	Activities	Best pChEMBL
CHEMBL182888	—	—	1	9.22

Activity Data

Compound	Name	Type	Rel.	Value	Units	pChEMBL
CHEMBL182888	—	IC50	=	0.6	nM	9.22