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Assay Detail

CHEMBL1220333

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Binding affinity to HCV 2AP54-labelled IRES subdomain 2a RNA in presence of 0.3 mM Mg2+ by FRET assay
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Hepacivirus hominis
Confidence 3 — Cell-line / Tissue
Curated By Autocuration

Target

Internal ribosome entry site (IRES) (CHEMBL612412)
Type NUCLEIC-ACID
Organism Hepacivirus hominis

Publication

Conformational inhibition of the hepatitis C virus internal ribosome entry site RNA.
Parsons J, Castaldi MP, Dutta S, Dibrov SM, Wyles DL, Hermann T.
Nat Chem Biol (2009) 5 : 823 -825
PubMed 19767736 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 1 6.58 6.58

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL223720 1 6.58

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL223720 EC50 = 260.0 nM 6.58