Assay Detail
Binding
CHEMBL1224955
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of Drosophila melanogaster SU(VAR)3-9
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Drosophila melanogaster |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Histone-lysine N-methyltransferase Su(var)3-9 (CHEMBL2169720) ↗| Type | SINGLE PROTEIN |
| Organism | Drosophila melanogaster |
Publication
Identification of a specific inhibitor of the histone methyltransferase SU(VAR)3-9.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 6.22 | 6.22 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1089316 | CHAETOCIN | — | 1 | 6.22 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1089316 | CHAETOCIN | IC50 | = | 600.0 | nM | 6.22 |