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Assay Detail

CHEMBL1243640

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Functional
Inhibition of 50 nM rapamycin-mediated cytostatic effect in yeast BY4742 after 48 to 96 hrs
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Saccharomyces cerevisiae
Confidence 1 — Organism
Curated By Autocuration

Target

Saccharomyces cerevisiae (CHEMBL361)
Type ORGANISM
Organism Saccharomyces cerevisiae

Publication

Small molecules enhance autophagy and reduce toxicity in Huntington's disease models.
Sarkar S, Perlstein EO, Imarisio S, Pineau S, Cordenier A, Maglathlin RL, Webster JA, Lewis TA, O'Kane CJ, Schreiber SL, Rubinsztein DC.
Nat Chem Biol (2007) 3 : 331 -338
PubMed 17486044 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 2 5.68 6.38

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL404954 1 6.38
CHEMBL312487 1 4.98

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL404954 EC50 = 412.0 nM 6.38
CHEMBL312487 EC50 = 10400.0 nM 4.98