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Assay Detail

CHEMBL1244642

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Binding affinity to human kallikrein 2
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Kallikrein-2 (CHEMBL2442)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Phage-encoded combinatorial chemical libraries based on bicyclic peptides.
Heinis C, Rutherford T, Freund S, Winter G.
Nat Chem Biol (2009) 5 : 502 -507
PubMed 19483697 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 5.47 5.47

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1240617 1 5.47

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1240617 IC50 = 3400.0 nM 5.47