Assay Detail
Functional
CHEMBL1249409
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Antiproliferative activity against human U2OS cells expressing constitutively active Stat3 mutant after 48 hrs by CMV-GFP reporter assay method
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | U2OS |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
A functional genomics approach to the mode of action of apratoxin A.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 7.30 | 7.30 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL501696 | APRATOXIN A | — | 1 | 7.30 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL501696 | APRATOXIN A | IC50 | = | 50.0 | nM | 7.30 |