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Assay Detail

CHEMBL1250107

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of v-Src kinase I338G mutant
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Target

Unchecked (CHEMBL612545)
Type UNCHECKED

Publication

Assignment of protein function in the postgenomic era.
Saghatelian A, Cravatt BF.
Nat Chem Biol (2005) 1 : 130 -142
PubMed 16408016 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 2 8.60 8.82

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL264406 1 8.82
CHEMBL573578 1 8.37

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL264406 IC50 = 1.5 nM 8.82
CHEMBL573578 IC50 = 4.3 nM 8.37