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Assay Detail

CHEMBL1263015

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiviral activity against Hepatitis B virus
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Hepatitis B virus
Confidence 1 — Organism
Curated By Autocuration

Target

Hepatitis B virus (CHEMBL613497)
Type ORGANISM
Organism Hepatitis B virus

Publication

Entecavir exhibits inhibitory activity against human immunodeficiency virus under conditions of reduced viral challenge.
Lin PF, Nowicka-Sans B, Terry B, Zhang S, Wang C, Fan L, Dicker I, Gali V, Higley H, Parkin N, Tenney D, Krystal M, Colonno R.
Antimicrob Agents Chemother (2008) 52 : 1759 -1767
PubMed 18316521 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 1 8.40 8.40

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL5314362 ENTECAVIR 4.0 1 8.40

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL5314362 ENTECAVIR EC50 = 4.0 nM 8.40