Assay Detail
Binding
CHEMBL1274081
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Inhibition of Penicillium decumbens naringinase after 10 to 30 mins
6
Total Activities
6
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Penicillium decumbens |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Fluorescent-tagged sp2-iminosugars with potent β-glucosidase inhibitory activity.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 6 | 6.48 | 7.14 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1272019 | — | — | 1 | 7.14 |
| CHEMBL1269790 | — | — | 1 | 6.75 |
| CHEMBL1272018 | — | — | 1 | 6.68 |
| CHEMBL1271962 | — | — | 1 | 6.64 |
| CHEMBL1269789 | — | — | 1 | 5.92 |
| CHEMBL1271963 | — | — | 1 | 5.75 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1272019 | — | Ki | = | 72.0 | nM | 7.14 |
| CHEMBL1269790 | — | Ki | = | 180.0 | nM | 6.75 |
| CHEMBL1272018 | — | Ki | = | 210.0 | nM | 6.68 |
| CHEMBL1271962 | — | Ki | = | 230.0 | nM | 6.64 |
| CHEMBL1269789 | — | Ki | = | 1200.0 | nM | 5.92 |
| CHEMBL1271963 | — | Ki | = | 1800.0 | nM | 5.75 |