Assay Detail
Binding
CHEMBL1282597
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Binding affinity to human recombinant GABA alpha-3-beta-2-gamma-2 receptor
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 7 — Homologous single protein target |
| Curated By | Intermediate |
Target
GABA A receptor alpha-3/beta-2/gamma-2 (CHEMBL2111339) ↗| Type | PROTEIN COMPLEX |
| Organism | Homo sapiens |
Publication
The GABA(A) receptor as a target for photochromic molecules.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 1 | 8.04 | 8.04 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL415290 | Ro-151310 | — | 1 | 8.04 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL415290 | Ro-151310 | Ki | = | 9.2 | nM | 8.04 |